DFG-1 Residue Controls Inhibitor Binding Mode and Affinity, Providing a Basis for Rational Design of Kinase Inhibitor Selectivity

Schröder M., Bullock AN., Fedorov O., Bracher F., Chaikuad A., Knapp S.

DOI

10.1021/acs.jmedchem.0c00898

Type

Journal article

Journal

Journal of Medicinal Chemistry

Publisher

American Chemical Society (ACS)

Publication Date

24/09/2020

Volume

63

Pages

10224 - 10234

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