Novel p38α MAP kinase inhibitors identified from yoctoReactor DNA-encoded small molecule library
Petersen LK., Blakskjær P., Chaikuad A., Christensen AB., Dietvorst J., Holmkvist J., Knapp S., Kořínek M., Larsen LK., Pedersen AE., Röhm S., Sløk FA., Hansen NJV.
<p>A DNA-encoded small-molecule library was prepared using yoctoReactor technology followed by binder trap enrichment to identify selective inhibitors with nanomolar potencies against p38α MAP kinase.</p>